www.bioscience.co.uk
Sales & Support: +44 (0)1223 316 855

*

Rilmenidine

Catalogue number:
CAY32879-1 g
Supplier:
Size:
1 g
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£1058.00 Estimated delivery Wed 24 Dec
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

54187-04-1

Purity:

≥95%

Formulation:

A crystalline solid

Molecular Formula:

C10H16N2O

Molecular Weight:

180.24692

Alternative Names:

n-(dicyclopropylmethyl)-4,5-dihydro-2-oxazolamine, nsc 664312, oxaminozoline

Product Description:

An antihypertensive agent; binds to imidazole receptors in bovine rostral ventrolateral medulla homogenates (Ki = 6.1 nM); binds α2-adrenergic receptors in bovine prefrontal cortex homogenates (Ki = 87 nM); induces hypotension and bradycardia in anesthetized rats (ED50s = 0.25 and 0.35 mg/kg, respectively); reduces mean arterial pressure and renal sympathetic nerve activity in a rabbit model of renal hypertension induced by a renal artery clip at 2.5 mg/kg; increases levels of LC3-II, a marker of autophagy, in PC12 cells at 1 µM