Dermorphin (acetate)
Catalogue number:
CAY31607-25 mg
Supplier:
Size:
25 mg
Product is available in:
£743.00
Estimated delivery Wed 11 Feb
Shipping is calculated in checkout
Shipping is calculated in checkout
Purity:
≥95%
Molecular Weight:
802.87292
Alternative Names:
(s)-1-(l-tyrosyl-
- MSDS: View or download
Product Description:
An opioid peptide; binds to µ-opioid receptors (Ki = 0.54 nM) and is selective for µ- over δ-opioid receptors in radioligand binding assays (Ki = 929 nM); inhibits noxious stimuli-induced neuronal firing in the nucleus lateralis anterior and ventrobasal complex in rats at 1.9 µmol/kg; inhibits the electrical stimulation-induced C fiber response in rat dorsal horn nociceptive neurons; delays gastric emptying, inhibits gastric acid secretion, and slows colonic motility in pylorus-ligated rats from 10-120 pmol/animal