AC-262536
Catalogue number:
CAY31598-10 mg
Supplier:
Size:
10 mg
Product is available in:
£432.00
Estimated delivery Wed 17 Dec
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
870888-46-3
Purity:
≥98%
Formulation:
A solid
Molecular Formula:
C18H18N2O
Molecular Weight:
278.4
Alternative Names:
4-[(3-endo)-
- MSDS: View or download
Product Description:
A SARM (Ki = 5.01 nM); an androgen receptor partial agonist (EC50 = 1.58 nM in a luciferase assay); selective for the androgen receptor over a panel of 47 additional human nuclear receptors at 10 µM; inhibits dihydroxytestosterone-induced proliferation of LNCaP prostate cancer cells at 0.1 and 1 µM; reduces plasma luteinizing hormone levels and increases levator ani muscle weight in castrated rats at 3, 10, and 30 mg/kg; exhibits smaller increases in prostate gland and seminal vesicle weight compared with testosterone in the same model