WM-1119
Catalogue number:
CAY30509-25 mg
Supplier:
Size:
25 mg
Product is available in:
£567.00
Estimated delivery Tue 26 May
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
2055397-28-7
Purity:
≥98%
Formulation:
A crystalline solid
Molecular Formula:
C18H13F2N3O3S
Molecular Weight:
389.4
Alternative Names:
3-fluoro-5-
Product Description:
An inhibitor of KAT6A (IC50 = 6.3 nM); binds to KAT6A (Kd = 2 nM); selective for KAT6A over KAT5 and KAT7 (Kds = 2,200 and 500 nM, respectively), as well as a panel of 159 additional targets at 1 and 10 µM; inhibits proliferation of EMRK1184 B cell lymphoma cells (IC50 = 0.25 µM); reduces tumor growth and spleen weight in a murine EMRK1184 model at 50 mg/kg four times per day