HA-1077 (hydrochloride)
Catalogue number:
CAY10010559-50 mg
Supplier:
Size:
50 mg _$$_
Product is available in:
£126.00
Estimated delivery Wed 29 May
Shipping is calculated in checkout
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
203911-27-7
Purity:
≥98%
Formulation:
A crystalline solid
Molecular Weight:
364.3
Alternative Names:
hexahydro-1-(5-isoquinolinylsulfonyl)-1h-1,4-diazepine, dihydrochloride, fasudil
- Data sheet: View or download
- MSDS: View or download
Product Description:
A potent inhibitor of ROCK2, PRK-2, MSK1, and MAPKAP-K1b with IC50 values of 1.9, 4, 5, and 15 µM, respectively; has been shown to reduce blood vessel constriction, decreases pulmonary arterial pressure, inhibit tumor angiogenesis, and improve insulin signaling in a diabetic rat model; drug forms are marketed for the treatment of pulmonary arterial hypertension and stable angina
Storage Temperature:
-20°C
