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PI-3065

Catalogue number:
CAY9002394-25 mg
Supplier:
Size:
25 mg _$$_
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£717.00 Estimated delivery Wed 29 May
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

955977-50-1

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

506.6

Alternative Names:

6-[[4-(cyclopropylmethyl)-1-piperazinyl]methyl]-2-(5-fluoro-1h-indol-4-yl)-4-(4-morpholinyl)-thieno[3,2-d]pyrimidine

Product Description:

A PI3K p110δ inhibitor (IC50 = 15 nM); greater than 100-fold selective for p110δ over p110ɑ, p110β, p110γ, DNA-PK, and mTOR; decreases tumor weight and inhibits metastasis in a 4T1 murine mammary carcinoma model at 75 mg/kg

Storage Temperature:

-20°C

CAY9002394-25 mg: PI-3065
CAY9002394-25 mg: PI-3065
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