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Bisindolylmaleimide I

Catalogue number:
CAY13298-25 mg
Supplier:
Size:
25 mg _$$_
Product is available in:
  • UK
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  • Rest of World
£492.00 Estimated delivery Wed 3 Jul
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

133052-90-1

Purity:

≥95%

Formulation:

A crystalline solid

Molecular Weight:

412.5

Alternative Names:

3-[1-[3-(dimethylamino)propyl]-1h-indol-3-yl]-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dione, bim i, gf 109203x, gö 6850

Product Description:

A highly selective, cell-permeable, and reversible PKC inhibitor (Ki = 14 nM); competitive inhibitor for the ATP binding site of PKC; highly selective for PKCα, β1, β2, γ, δ, and ε isozymes; inhibits GSK3 in primary adipocyte lysates (IC50 = 360 nM) and in GSK3β immunoprecipitates derived from rat epididymal adipocytes (IC50 = 170 nM); competitively antagonizes the 5-HT3 receptor with a Ki value of 61 nM

Storage Temperature:

-20°C

Details Cat number & supplier Size Price
Bisindolylmaleimide I (hydrochloride) CAY21180-1 mg · Cayman Chemical
CAY21180-1 mg
Cayman Chemical
1 mg £65.00
1 mg
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