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FK-866

Catalogue number:
CAY13287-25 mg
Supplier:
Size:
25 mg _$$_
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£455.00 Estimated delivery Tue 21 May
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

658084-64-1

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

391.5

Alternative Names:

n-[4-(1-benzoyl-4-piperidinyl)butyl]-3-(3-pyridinyl)-2e-propenamide, ​daporinad, apo-866, k 22.175

Product Description:

A highly specific non-competitive inhibitor of Nampt (Ki = 0.4 nM), causing gradual NAD+ depletion; directs delayed cell death by apoptosis in HepG2 cells (IC50 = ~1 nM)

Storage Temperature:

-20°C

CAY13287-25 mg: FK-866
CAY13287-25 mg: FK-866
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