£238.00
Estimated delivery Wed 15 May
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
155270-99-8
Purity:
≥98%
Formulation:
A crystalline solid
Molecular Weight:
384.4
Alternative Names:
8-[(1e)-2-(3,4-dimethoxyphenyl)ethenyl]-1,3-diethyl-3,7-dihydro-7-methyl-1h-purine-2,6-dione, kw 6002
- Data sheet: View or download
- MSDS: View or download
Product Description:
An A2A receptor antagonist (Ki = 2.2 nM in a radioligand binding assay); inhibits haloperidol-induced catalepsy (ED50 = 0.23 mg/kg in rats); alleviates postural defects in a dose-dependent manner without inducing dyskinesias or hyperactivity in an MPTP-induced marmoset model of Parkinson's disease; decreases bradykinesias induced by L-DOPA and improves attentional and working memory deficits in an MPTP-induced macaque model of Parkinson's disease
Storage Temperature:
-20°C