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NCT-503

Catalogue number:
CAY19718-1 mg
Supplier:
Size:
1 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£42.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1916571-90-8

Purity:

≥98%

Formulation:

A neat solid

Molecular Weight:

408.5

Alternative Names:

n-(4,6-dimethyl-2-pyridinyl)-4-[[4-(trifluoromethyl)phenyl]methyl]-1-piperazinecarbothioamide

Product Description:

A PHGDH inhibitor that blocks serine synthesis from 3-phosphoglycerate in cells (IC50 = 2.5 µM); reduces the production of glucose-derived serine in cells and suppresses the growth of PHGDH-dependent MDA-MB-468 cancer cells both in vitro and in mice bearing orthotopic xenograft tumors

Storage Temperature:

-20°C

CAY19718-1 mg: NCT-503
CAY19718-1 mg: NCT-503
Details Cat number & supplier Size Price
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NCT-503 CAY19718-10 mg · Cayman Chemical
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PHGDH-inactive CAY19717-25 mg · Cayman Chemical
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NCT-503 CAY19718-25 mg · Cayman Chemical
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PHGDH-inactive CAY19717-10 mg · Cayman Chemical
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10 mg £493.00
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NCT-503 CAY19718-5 mg · Cayman Chemical
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5 mg £112.00
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PHGDH-inactive CAY19717-1 mg · Cayman Chemical
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GSK583 CAY19739-100 mg · Cayman Chemical
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