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BIIB021

Catalogue number:
CAY18269-5 mg
Supplier:
Size:
5 mg _$$_
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£65.00 Estimated delivery Tue 14 May
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

848695-25-0

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

318.8

Alternative Names:

6-chloro-9-[(4-methoxy-3,5-dimethyl-2-pyridinyl)methyl]-9h-purin-2-amine, cnf2024

Product Description:

A potent, orally-available inhibitor of Hsp90 (Ki = 1.7 nM) that induces the degradation of oncoproteins, including HER2 (EC50 = 38 nM), while up-regulating the expression of Hsp70 and Hsp27; cytotoxic to cancer cells and, when administered orally to mice, inhibits growth of xenograft tumors

Storage Temperature:

-20°C

CAY18269-5 mg: BIIB021
CAY18269-5 mg: BIIB021
Details Cat number & supplier Size Price
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