www.bioscience.co.uk
Sales & Support: +44 (0)1223 316 855

*

MK-0457

Catalogue number:
CAY13600-50 mg
Supplier:
Size:
50 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£209.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

639089-54-6

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

464.6

Alternative Names:

n-[4-[[4-(4-methyl-1-piperazinyl)-6-[(5-methyl-1h-pyrazol-3-yl)amino]-2-pyrimidinyl]thio]phenyl]-cyclopropanecarboxamide, tozasertib, vx-680

Product Description:

A potent pan-Aurora kinase inhibitor that favors Aurora A (Ki = 0.6 nM) over Aurora B (Ki = 18 nM) or Aurora C (Ki = 4.6 nM); inhibits proliferation of clear cell renal carcinoma (IC50 = 2/M phase

Storage Temperature:

-20°C

CAY13600-50 mg: MK-0457
CAY13600-50 mg: MK-0457
Details Cat number & supplier Size Price
JNJ-26854165 CAY16259-10 mg · Cayman Chemical
CAY16259-10 mg
Cayman Chemical
10 mg £277.00
10 mg
view
(R)-CR8 CAY14006-10 mg · Cayman Chemical
CAY14006-10 mg
Cayman Chemical
10 mg £433.00
10 mg
view
MJ33 (lithium salt) CAY90001844-5 mg · Cayman Chemical
CAY90001844-5 mg
Cayman Chemical
5 mg £209.00
5 mg
view
Lanicemine CAY9002129-10 mg · Cayman Chemical
CAY9002129-10 mg
Cayman Chemical
10 mg £124.00
10 mg
view
Quetiapine (hemifumarate) CAY14152-10 g · Cayman Chemical
CAY14152-10 g
Cayman Chemical
10 g £278.00
10 g
view
Indoxyl Sulfate (potassium salt) CAY16926-1 g · Cayman Chemical
CAY16926-1 g
Cayman Chemical
1 g £204.00
1 g
view
R-59-022 CAY16772-10 mg · Cayman Chemical
CAY16772-10 mg
Cayman Chemical
10 mg £204.00
10 mg
view
Enoxacin CAY16956-5 g · Cayman Chemical
CAY16956-5 g
Cayman Chemical
5 g £278.00
5 g
view
5-Octyl-α-ketoglutarate CAY16105-1 mg · Cayman Chemical
CAY16105-1 mg
Cayman Chemical
1 mg £117.00
1 mg
view
Biotin-azide CAY13040-5 mg · Cayman Chemical
CAY13040-5 mg
Cayman Chemical
5 mg £216.00
5 mg
view