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LGK974

Catalogue number:
CAY14072-1 mg
Supplier:
Size:
1 mg _$$_
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£89.00 Estimated delivery Wed 15 May
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1243244-14-5

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

396.4

Alternative Names:

2',3-dimethyl-n-[5-(2-pyrazinyl)-2-pyridinyl]-[2,4'-bipyridine]-5-acetamide, porcn inhibitor iv

Product Description:

A potent and specific small molecule inhibitor of PORCN (IC50 = 0.4 nM); greatly reduces Wnt secretion without decreasing its synthesis and without increasing cytotoxicity; orally bioavailable in mice

Storage Temperature:

-20°C

CAY14072-1 mg: LGK974
CAY14072-1 mg: LGK974
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