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OTX015

Catalogue number:
CAY15947-1 mg
Supplier:
Size:
1 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£64.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

202590-98-5

Purity:

≥95%

Formulation:

A crystalline solid

Molecular Weight:

492

Alternative Names:

(6s)-4-(4-chlorophenyl)-n-(4-hydroxyphenyl)-2,3,9-trimethyl-6h-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetamide, (−)-otx015, hy-15743

Product Description:

An orally bioavailable, small molecule inhibitor of BRD2, BRD3, and BRD4 (EC50s = 10-19 nM) that displays antiproliferative effects at a sub-micromolar range in vitro in a wide range of solid tumor types and leukemias

Storage Temperature:

-20°C

CAY15947-1 mg: OTX015
CAY15947-1 mg: OTX015
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