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BRD0639

Catalogue number:
CAY35625-1 mg
Supplier:
Size:
1 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£125.00 Estimated delivery Wed 7 Aug
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
Purity:

≥98%

Formulation:

A solid

Molecular Weight:

475.9

Alternative Names:

(s)-2-(4-chloro-6-oxopyridazin-1(6h)-yl)-n-(4-methyl-3-(n-(2-(pyridin-2-yl)ethyl)sulfamoyl)phenyl)propanamide

Product Description:

An inhibitor of the protein-peptide interaction between PRMT5 and PBM (IC50 = 13.8 µM); induces the formation of PRMT5 adducts in cells (EC50 = 3 µM) and disrupts complex formation between PRMT5 and RIOK1 in permeabilized cells

Storage Temperature:

-20°C

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