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SR 144528

Catalogue number:
CAY9000491-25 mg
Supplier:
Size:
25 mg _$$_
Product is available in:
  • UK
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£676.00 Estimated delivery Wed 31 Jul
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

192703-06-3

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

476.1

Alternative Names:

5-(4-chloro-3-methylphenyl)-1-[(4-methylphenyl)methyl]-n-[(1s,2s,4r)-1,3,3-trimethylbicyclo[2.2.1]hept-2-yl]-1h-pyrazole-3-carboxamide

Product Description:

A CB2 receptor antagonist (Ki = 0.6 nM); selective for CB2 over CB1 receptors in CHO cells expressing human receptors (Ki = 437 nM); reverses CP 55,940-induced inhibition of forskolin-induced adenylyl cyclase activity in CHO cells expressing human CB2 receptors (EC50 = 10 nM); reduces paw swelling in a mouse model of carrageenin-induced paw edema at 0.01 mg/kg

Storage Temperature:

-20°C

CAY9000491-25 mg: SR 144528
CAY9000491-25 mg: SR 144528
Details Cat number & supplier Size Price
SR 144528-d3 CAY37830-500 ug · Cayman Chemical
CAY37830-500 ug
Cayman Chemical
500 µg £213.00
500 µg
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