GSK 1016790A
Catalogue number:
B2952-25
Supplier:
BioVision
Size:
25 mg _$$_
Product is available in:
N/A
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CAS Number:
942206-85-1
Purity:
98%
Molecular Weight:
655
Alternative Names:
N-[(2S)-1-[4-[(2S)-2-[(2,4-dichlorophenyl)sulfonylamino]-3-hydroxypropanoyl]piperazin-1-yl]-4-methyl-1-oxopentan-2-yl]-1-benzothiophene-2-carboxamide; N-[(1S)-1-[[4-[(2S)-2-[[(2,4-dichlorophenyl)sulfonyl]amino]-3-hydroxy-1-oxopropyl]-1-piperazinyl]carbony
- Data sheet: View or download
- MSDS: View or download
Product Description:
GSK1016790A is a transient receptor potential vanilloid 4 (TRPV4) agonist that elicits calcium influx in HEK cells expressing mouse or human transient TRPV4 with EC₅₀ values of 18 and 2.1 nM, respectively. It regulates urinary bladder activity and infusion of GSK1016790A into the bladders of TRPV4+/+ mice induces bladder overactivity.
Storage Temperature:
-20°C