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GSK 1016790A

Catalogue number:
Supplier:
BioVision
Size:
25 mg _$$_
Product is available in:
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CAS Number:

942206-85-1

Purity:

98%

Molecular Weight:

655

Alternative Names:

N-[(2S)-1-[4-[(2S)-2-[(2,4-dichlorophenyl)sulfonylamino]-3-hydroxypropanoyl]piperazin-1-yl]-4-methyl-1-oxopentan-2-yl]-1-benzothiophene-2-carboxamide; N-[(1S)-1-[[4-[(2S)-2-[[(2,4-dichlorophenyl)sulfonyl]amino]-3-hydroxy-1-oxopropyl]-1-piperazinyl]carbony

Product Description:

GSK1016790A is a transient receptor potential vanilloid 4 (TRPV4) agonist that elicits calcium influx in HEK cells expressing mouse or human transient TRPV4 with EC₅₀ values of 18 and 2.1 nM, respectively. It regulates urinary bladder activity and infusion of GSK1016790A into the bladders of TRPV4+/+ mice induces bladder overactivity.

Storage Temperature:

-20°C

GSK 1016790A
GSK 1016790A