www.bioscience.co.uk
Sales & Support: +44 (0)1223 316 855

*

XMD17-109

Supplier:
Catalogue number:
CAY25448-25 mg
Size:
25 mg
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£486.00 Estimated delivery Tue 4 May
Shipping is calculated in checkout

A selective ERK5 inhibitor (IC50 = 0.162 µM in an enzyme assay); selective for ERK5 over a panel of more than 200 kinases at 10 µM; inhibits ERK5 phosphorylation (IC50 = 0.09 µM in HeLa cells); decreases AP-1 transcriptional activity (EC50 = 4.2 µM); inhibits human recombinant LRRK2[G2019S] (IC50 = 0.339 µM in an enzyme assay)

Product Type:

Biochemicals

CAS Number:

1435488-37-1

Alternative Names:

11-cyclopentyl-2-[[2-ethoxy-4-[[4-(4-methyl-1-piperazinyl)-1-piperidinyl]carbonyl]phenyl]amino]-5,11-dihydro-5-methyl-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one, erk5-in-1

Storage Temp:

-20°C

Formulation:

A crystalline solid

Compound Purity:

≥98%

UNSPSC Code:

12352200

CAY25448-25 mg: XMD17-109

CAY25448-25 mg: XMD17-109