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XMD17-109

Catalogue number:
CAY25448-25 mg
Supplier:
Size:
25 mg _$$_
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£616.00 Estimated delivery Tue 9 Apr
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1435488-37-1

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

638.8

Alternative Names:

11-cyclopentyl-2-[[2-ethoxy-4-[[4-(4-methyl-1-piperazinyl)-1-piperidinyl]carbonyl]phenyl]amino]-5,11-dihydro-5-methyl-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one, erk5-in-1

Product Description:

A selective ERK5 inhibitor (IC50 = 0.162 µM in an enzyme assay); selective for ERK5 over a panel of more than 200 kinases at 10 µM; inhibits ERK5 phosphorylation (IC50 = 0.09 µM in HeLa cells); decreases AP-1 transcriptional activity (EC50 = 4.2 µM); inhibits human recombinant LRRK2[G2019S] (IC50 = 0.339 µM in an enzyme assay)

Storage Temperature:

-20°C

CAY25448-25 mg: XMD17-109
CAY25448-25 mg: XMD17-109
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