VU0364572 (trifluoroacetate salt)
Catalogue number:
CAY20466-25 mg
Supplier:
Size:
25 mg _$$_
Product is available in:
£1295.00
Estimated delivery Tue 30 Apr
Shipping is calculated in checkout
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
1240514-89-9
Purity:
≥98%
Formulation:
A crystalline solid
Molecular Weight:
487.5
Alternative Names:
(3r)-3-[(2-methylbenzoyl)amino]-[1,4'-bipiperidine]-1'-carboxylic acid, ethyl ester, 2,2,2-trifluoroacetate
- Data sheet: View or download
- MSDS: View or download
Product Description:
A potent and selective agonist of M1 receptors (EC50 = 0.2 mM compared to >10 mM for M2-M5); induces concentration-dependent increases in Ca2+ mobilization and ERK1/2 phosphorylation in hM1 CHO cells (EC50s = 0.89 and 10 mM, respectively); improves hippocampal-dependent spatial learning and localization abilities and acquistion of contextual fear learning but cannot reverse amphetamine-induced hyperlocamotion in rats
Storage Temperature:
-20°C