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PCNA-I1

Catalogue number:
CAY20454-25 mg
Supplier:
Size:
25 mg _$$_
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£392.00 Estimated delivery Tue 9 Apr
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

444930-42-1

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

310.4

Alternative Names:

3-methyl-2-[(1-hydroxy-2-naphthalenyl)methylene]hydrazide-2-thiophenecarboxylic acid

Product Description:

An inhibitor of PCNA; binds to PCNA trimers (Kd = 0.41 µM) and reduces the level of chromatin-associated PCNA in PC3 cells; preferentially inhibits growth of a variety of human and mouse cancer cell lines (IC50s = 0.05-0.3 µM) over non-transformed cells (IC50s = 0.99-2 µM); reduces tumor growth in an LNCaP prostate cancer mouse xenograft model at 10 mg/kg administered five days per week for two weeks

Storage Temperature:

-20°C

CAY20454-25 mg: PCNA-I1
CAY20454-25 mg: PCNA-I1
Details Cat number & supplier Size Price
PCNA-I1 CAY20454-5 mg · Cayman Chemical
CAY20454-5 mg
Cayman Chemical
5 mg £89.00
5 mg
view
PCNA-I1 CAY20454-10 mg · Cayman Chemical
CAY20454-10 mg
Cayman Chemical
10 mg £169.00
10 mg
view
PCNA-I1 CAY20454-50 mg · Cayman Chemical
CAY20454-50 mg
Cayman Chemical
50 mg £694.00
50 mg
view
LDN-211904 CAY20453-5 mg · Cayman Chemical
CAY20453-5 mg
Cayman Chemical
5 mg £284.00
5 mg
view
OXA-01 CAY20456-1 mg · Cayman Chemical
CAY20456-1 mg
Cayman Chemical
1 mg £42.00
1 mg
view
OXA-01 CAY20456-10 mg · Cayman Chemical
CAY20456-10 mg
Cayman Chemical
10 mg £299.00
10 mg
view
LDN-211904 CAY20453-1 mg · Cayman Chemical
CAY20453-1 mg
Cayman Chemical
1 mg £89.00
1 mg
view
OXA-01 CAY20456-25 mg · Cayman Chemical
CAY20456-25 mg
Cayman Chemical
25 mg £691.00
25 mg
view
Madrasin CAY20451-5 mg · Cayman Chemical
CAY20451-5 mg
Cayman Chemical
5 mg £121.00
5 mg
view
OXA-01 CAY20456-5 mg · Cayman Chemical
CAY20456-5 mg
Cayman Chemical
5 mg £181.00
5 mg
view