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CAS Number:
183232-66-8
Purity:
≥98%
Molecular Weight:
555
Alternative Names:
1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-N-1-piperidinyl-1H-pyrazole-3-carboxamide,AM251
- Data sheet: View or download
- MSDS: View or download
Product Description:
AM251 is a selective cannabinoid 1 (CB1) receptor antagonist with an IC50 of 8 nM. It also acts as an agonist at GPR55 (EC50 = 39 nM) and potentiates GABAA receptor currents (EC50 = 0.4 µM). In mice, AM251 reduces antidepressant-like behavior in the tail suspension and forced swim tests and decreases hyperphagia induced by fasting.
Storage Temperature:
-20°C
