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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
5588-33-0
Purity:
≥95%
Formulation:
A solution in acetonitrile
Molecular Weight:
386.6
Alternative Names:
10-[2-(1-methyl-2-piperidinyl)ethyl]-2-(methylsulfinyl)-10h-phenothiazine, nsc 186066
Product Description:
An active metabolite of thioridazine; formed via sulfoxidation of thioridazine by CYP2D6 in human liver microsomes; binds to histamine H1, dopamine D2, muscarinic acetylcholine, and α1- and α2-adrenergic receptors (Kds = 1.8, 19, 69, 2, and 1,600 nM, respectively); prevents mescaline-induced hyperactivity in mice at 10, 30, and 45 mg/kg
Storage Temperature:
-20°C