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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
2854-32-2
Purity:
≥98%
Formulation:
A crystalline solid
Molecular Weight:
426.9
Alternative Names:
2-[1-(4-chlorobenzoyl)-5-methoxy-2-methyl-1h-indol-3-yl]-1-(4-morpholinyl)-ethanone, bml-190, indomethacin morpholinylamide, lm-4131
- Data sheet: View or download
- MSDS: View or download
Product Description:
A CB2 receptor inverse agonist (Ki = 435 nM for recombinant human CB2); selective for CB2 over CB1 receptors (Ki = >20 µM); reduces basal production of inositol phosphate and increases forskolin-induced accumulation of cAMP in HEK293 cells expressing human CB2 receptors from 0.001-1 µM; inhibits LPS-induced NO and PGE2 production in J774 macrophages
Storage Temperature:
-20°C