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PF-04937319 (hydrate)

Catalogue number:
CAY30926-10 mg
Supplier:
Size:
10 mg _$$_
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£253.00 Estimated delivery Tue 7 May
Shipping is calculated in checkout
Purity:

≥98%

Molecular Weight:

432.4

Alternative Names:

n,n-dimethyl-5-[[2-methyl6-[[5-methyl-2-pyrazinyl)amino]carbonyl]-4-benzofuranyl]oxy]-2-pyrimidinecarboxamide, hydrate

Product Description:

A glucokinase activator (EC50s = 174, 407, and 269 nM for the recombinant human, rat, and dog enzymes, respectively); increases glucose-induced insulin secretion in isolated rat islets at 4 and 12 µM; reduces postprandial plasma glucose levels in rats from 3-100 mg/kg

Storage Temperature:

-20°C

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