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eCF506

Catalogue number:
CAY19959-25 mg
Supplier:
Size:
25 mg _$$_
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£414.00 Estimated delivery Tue 9 Apr
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1914078-41-3

Purity:

≥98%

Formulation:

A crystalline solid

Molecular Weight:

510.6

Alternative Names:

n-[4-[4-amino-1-[2-[4-(dimethylamino)-1-piperidinyl]ethyl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl]-2-methoxyphenyl]-carbamic acid, 1,1-dimethylethyl ester

Product Description:

An inhibitor of Src kinases (IC50s = 50 = 479 nM), as well as KIT, mTOR, PDGFRα, and RET (IC50s = >100 µM for all); completely inhibits Src and FAK phosphorylation at 100 nM; inhibits proliferation of MCF-7 cells (EC50 = 9 nM); reduces levels of activated Src kinase in tumor tissue in an HCT116 mouse xenograft model at 50 mg/kg per day

Storage Temperature:

-20°C

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