Mitiglinide (calcium salt)
Catalogue number:
CAY30693-500 mg
Supplier:
Size:
500 mg _$$_
Product is available in:
£601.00
Estimated delivery Wed 1 May
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
145525-41-3
Purity:
≥98% (mixture of isomers)
Formulation:
A crystalline solid
Molecular Weight:
334.4
Alternative Names:
(αs,3ar,7as)-octahydro-γ-oxo-α-(phenylmethyl)-2h-isoindole-2-butanoic acid, hemicalcium salt, kad-1229, s21403
- Data sheet: View or download
- MSDS: View or download
Product Description:
A SUR1/Kir6.2 inhibitor (IC50 = 4 nM); selective for SUR1/Kir6.2 over SUR2A/Kir6.2 and SUR2B/Kir6.2 channels (IC50s = 3 and 5 µM, respectively); induces insulin release in HIT-T15 insulinoma cells and isolated mouse pancreatic islets at 100 µM; increases postprandial plasma insulin levels and inhibits postprandial increases in plasma glucose levels in an STZ-induced rat model of diabetes
Storage Temperature:
-20°C