www.bioscience.co.uk
Sales & Support: +44 (0)1223 316 855

*

ERGi-USU

Catalogue number:
CAY30875-1 g
Supplier:
Size:
1 g _$$_
Product is available in:
  • UK
  • Ireland
  • Europe
  • USA
  • Rest of World
£247.00 Estimated delivery Tue 9 Apr
Shipping is calculated in checkout
This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:

1147-56-4

Purity:

≥98%

Formulation:

A solid

Molecular Weight:

255.3

Alternative Names:

1-[2-(2-thiazolyl)diazenyl]-2-naphthalenol, nsc 139021

Product Description:

An ERG inhibitor (IC50 = 315 nM); inhibits proliferation of ERG-expressing VCaP prostate, COLO 320 colon, and KG-1 and MOLT-4 leukemia cancer cells (IC50s = 30-400 nM) but LNCaP, LAPC4, and MDA PCa 2b prostate cancer and HUVECs, which do not express ERG (IC50s = >10 µM for all); reduces tumor growth in a VCaP mouse xenograft model at 100 and 150 mg/kg

Storage Temperature:

-20°C

Details Cat number & supplier Size Price
Takinib CAY24161-5 mg · Cayman Chemical
CAY24161-5 mg
Cayman Chemical
5 mg £112.00
5 mg
view
ERGi-USU CAY30875-100 mg · Cayman Chemical
CAY30875-100 mg
Cayman Chemical
100 mg £59.00
100 mg
view
Takinib CAY24161-25 mg · Cayman Chemical
CAY24161-25 mg
Cayman Chemical
25 mg £445.00
25 mg
view
ERGi-USU CAY30875-50 mg · Cayman Chemical
CAY30875-50 mg
Cayman Chemical
50 mg £43.00
50 mg
view
Takinib CAY24161-10 mg · Cayman Chemical
CAY24161-10 mg
Cayman Chemical
10 mg £199.00
10 mg
view
ERGi-USU CAY30875-500 mg · Cayman Chemical
CAY30875-500 mg
Cayman Chemical
500 mg £186.00
500 mg
view
Takinib CAY24161-1 mg · Cayman Chemical
CAY24161-1 mg
Cayman Chemical
1 mg £42.00
1 mg
view
SR 3576 CAY20215-1 mg · Cayman Chemical
CAY20215-1 mg
Cayman Chemical
1 mg £42.00
1 mg
view
ATRA-BA Hybrid CAY30982-5 mg · Cayman Chemical
CAY30982-5 mg
Cayman Chemical
5 mg £181.00
5 mg
view
SR 3576 CAY20215-5 mg · Cayman Chemical
CAY20215-5 mg
Cayman Chemical
5 mg £151.00
5 mg
view