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PF-05105679

Supplier:
Catalogue number:
CAY29489-1 mg
Size:
1 mg
Product is available in:
  • UK
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£32.00 Estimated delivery Fri 18 Jun
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A TRPM8 antagonist (IC50 = 103 nM for inhibition of voltage-activated currents in HEK293 cells expressing the human receptor); >100-fold selective for TRPM8 over a panel of 90 receptors, ion channels, and enzymes; inhibits cold- and WS-12-induced calcium flux in HEK293 cells expressing the human TRPM8 (IC50s = 480 and 181 nM, respectively); reverses cold-induced reductions in bladder capacity in anesthetised guinea pigs when administered as an i.v. infusion at 46.67 µg/kg per minute; decreases the core body temperature in rats at 100 and 300 mg/kg

Product Type:

Biochemicals

CAS Number:

1398583-31-7

Alternative Names:

3-[[[(1r)-1-(4-fluorophenyl)ethyl](3-quinolinylcarbonyl)amino]methyl]-benzoic acid

Storage Temp:

-20°C

Formulation:

A solid

Compound Purity:

≥98%

UNSPSC Code:

12352200

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