£81.00
Estimated delivery Wed 15 May
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This product is for research use only and is not for human consumption or therapeutic use.
CAS Number:
865362-74-9
Purity:
≥98%
Formulation:
A crystalline solid
Molecular Weight:
327.3
Alternative Names:
5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridazin-3-amine, erk inhibitor ii
- Data sheet: View or download
- MSDS: View or download
Product Description:
A potent cell-permeable inhibitor of ERK1 and ERK2 (Ki = 310 and 140 nM, respectively); much less effective against p38α (IC50 = 10 µM) and does not inhibit a range of other serine/threonine or tyrosine kinases; blocks ERK-mediated signaling from TGF-β to AP-1 (IC50 = 3.1 µM)
Storage Temperature:
-20°C
